SCHEMBL9926386

SCHEMBL9926386

COCCN(C)Cc1csc2nc(-c3ccccc3NC(=O)c3ccc(OC)c(OC)c3)cn12

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 11/20 0.57
ABCG2 Q9UNQ0 3/20 0.44
MAPK1 P28482 1/20 0.44
PKM P14618 1/20 0.44
ABCB1 P08183 2/20 0.42
PDE4D Q08499 1/20 0.42
PDCD1 Q15116 1/20 0.42
CD274 Q9NZQ7 1/20 0.42
CHEK1 O14757 1/20 0.41
PIM1 P11309 1/20 0.41
MAPK8 P45983 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2624434 0.91 SIRT1 (0.60) SIRT1ABCG2MAPK1ABCB1PDE4D
SCHEMBL2624690 0.83 SIRT1 (0.72) SIRT1
SCHEMBL2624435 0.80 SIRT1 (0.71) SIRT1MAPK1PDCD1CD274
SCHEMBL2624433 0.80 SIRT1 (0.85) SIRT1ABCG2MAPK1ABCB1PDE4D
SCHEMBL2624436 0.75 SIRT1 (0.50) SIRT1ABCG2PKMABCB1PDE4D
SCHEMBL2624513 0.74 SIRT1 (0.87) SIRT1
SCHEMBL2624432 0.74 TP53 (0.69) SIRT1ABCG2MAPK1PKMABCB1
SCHEMBL2740381 0.74 SIRT1 (0.80) SIRT1CHEK1
SCHEMBL2740427 0.73 SIRT1 (0.68) SIRT1MAPK1
SCHEMBL20893167 0.72 SIRT1 (0.88) SIRT1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1955077-B1 MASS SPECTROMETRY ASSAYS FOR ACETYLTRANSFERASE/DEACETYLASE ACTIVITY SIRTRIS PHARMACEUTICALS INC (US) 2012-06-13 EP disclosed