SCHEMBL992893

SCHEMBL992893

CC(O)c1cccc2nc(-c3cc(-c4cnn(C)c4)cnc3N)[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MET P08581 5/20 0.49
LRRK2 Q5S007 3/20 0.45
CDK1 P06493 2/20 0.44
CDK2 P24941 2/20 0.44
MKNK1 Q9BUB5 2/20 0.44
MKNK2 Q9HBH9 2/20 0.44
PDPK1 O15530 1/20 0.44
MAP4K4 O95819 1/20 0.44
MAPK1 P28482 7/20 0.41
EPHX2 P34913 1/20 0.40
PIK3CD O00329 1/20 0.39
PIK3CB P42338 1/20 0.39
MTOR P42345 1/20 0.39
PIK3CG P48736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2680242 0.85 MET (0.53) METLRRK2CDK1CDK2MKNK1
SCHEMBL2680541 0.84 MET (0.53) METLRRK2CDK1CDK2MKNK1
SCHEMBL4088788 0.83 MET (0.50) METLRRK2CDK1CDK2MKNK1
SCHEMBL992891 0.82 MET (0.48) METLRRK2CDK1CDK2MKNK1
SCHEMBL2680942 0.79 CDK1 (0.70) METLRRK2CDK1CDK2MKNK1
SCHEMBL1045915 0.76 MAP4K4 (0.52) METLRRK2MAP4K4MAPK1
SCHEMBL2681519 0.75 LRRK2 (0.51) METLRRK2CDK1CDK2MKNK1
SCHEMBL16390689 0.75 LRRK2 (0.46) METLRRK2CDK1CDK2MKNK1
SCHEMBL2680902 0.75 MET (0.44) METLRRK2CDK1CDK2MKNK1
SCHEMBL4253781 0.75 CDK1 (0.52) METLRRK2CDK1CDK2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2454253-A1 AMINOPYRIDINE DERIVATIVES FOR TREATING TUMORS AND INFLAMMATORY DISEASES Merck Patent GmbH (DE) 2012-05-23 EP disclosed
WO-2011006567-A1 AMINOPYRIDINE DERIVATIVES FOR TREATING TUMORS AND INFLAMMATORY DISEASES MERCK PATENT GMBH (DE) 2011-01-20 WO disclosed