SCHEMBL9938053

SCHEMBL9938053

COC(=O)c1cc(C)c(S(=O)(=O)NC[C@H]2O[C@H](O)[C@@H](NC(=O)c3cccc(Br)c3)[C@@H](O)[C@@H]2O)s1

nearest known ligand 0.71

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HK2 P52789 17/20 0.71
HK1 P19367 16/20 0.71
GCK P35557 1/20 0.50
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LGALS9 O00182 1/20 0.36
LGALS8 O00214 1/20 0.36
LGALS1 P09382 1/20 0.36
LGALS3 P17931 1/20 0.36
LGALS7; LGALS7B P47929 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9938050 1.00 HK2 (0.71) HK2HK1GCKKDM4EALDH1A1
SCHEMBL9937446 0.69 HK1 (1.00) HK2HK1GCK
SCHEMBL9938423 0.68 HK2 (0.80) HK2HK1GCK
SCHEMBL4607774 0.67 MCL1 (0.46) ALDH1A1LMNA
SCHEMBL9937688 0.62 HK1 (0.69) HK2HK1GCKLMNAPOLB
SCHEMBL9937695 0.62 HK1 (0.69) HK2HK1GCKLMNAPOLB
SCHEMBL9938663 0.61 HK1 (0.73) HK2HK1GCK
SCHEMBL15881071 0.61 MCL1 (0.53) KDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL9938774 0.61 HK1 (0.60) HK2HK1GCKKDM4EALDH1A1
SCHEMBL9971331 0.60 HK1 (0.73) HK2HK1GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083145-A1 GLUCOSAMINE DERIVATIVES GLAXO WELLCOME MANUFACTURING PTE LTD (SG) 2012-06-21 WO disclosed