SCHEMBL9939494

SCHEMBL9939494

COc1ccc2c(F)[c]ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
CYP2A6 P11509 1/20 0.42
TRPA1 O75762 1/20 0.40
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.39
CYP3A4 P08684 1/20 0.39
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21830459 0.80 CYP1A2 (0.44) CYP1A2CYP2A6KDM4EMEN1MAPT
SCHEMBL6891247 0.79 CYP1A2 (0.42) CYP1A2CYP2A6KDM4EMEN1MAPT
SCHEMBL9365805 0.79 CYP1A2 (0.42) CYP1A2CYP2A6KDM4EMEN1MAPT
SCHEMBL7041458 0.78
SCHEMBL4079928 0.75 ALDH1A1 (0.42) CYP1A2CYP2A6KDM4EMEN1MAPT
SCHEMBL9939717 0.75 NQO1 (0.44) CYP1A2CYP2A6KDM4EMEN1MAPT
SCHEMBL25784076 0.74 CYP1A2 (0.50) CYP1A2CYP2A6TRPA1KDM4EMEN1
SCHEMBL1392528 0.74
SCHEMBL27902298 0.74 CYP2A6 (0.65) CYP1A2CYP2A6KDM4EMEN1MAPT
SCHEMBL3137389 0.72 CYP2A6 (0.62) CYP1A2CYP2A6KDM4EMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651871-A1 NOVEL SUBSTITUTED BICYCLIC AROMATIC COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS N30 Pharmaceuticals, Inc. (US) 2013-10-23 EP disclosed
WO-2012170371-A1 COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS N30 PHARMACEUTICALS, LLC (US) 2012-12-13 WO disclosed
WO-2012083171-A1 NOVEL SUBSTITUTED BICYCLIC AROMATIC COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS N30 PHARMACEUTICALS, LLC (US) 2012-06-21 WO disclosed