SCHEMBL9941215

SCHEMBL9941215

O=C(O)CN1CN(Cc2nc3cc(Cl)ccc3n2CCCCF)C2CN=CC=C21

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 9/20 0.38
BACE1 P56817 5/20 0.34
NUDT1 P36639 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9941216 0.74 TBXA2R (0.37) TBXA2R
SCHEMBL9979854 0.71 BACE1 (0.54) TBXA2RBACE1NUDT1KDM4EALDH1A1
SCHEMBL9979855 0.70 BACE1 (0.49) TBXA2RBACE1NUDT1
SCHEMBL9940520 0.69 CYP3A4 (0.45) TBXA2RKDM4EALDH1A1
Hydrochloric Acid SCHEMBL15301119 0.69 BACE1 (0.48) TBXA2RBACE1NUDT1
SCHEMBL23100606 0.67 MAPT (0.53) TBXA2RBACE1NUDT1
SCHEMBL9940732 0.63 CYP3A4 (0.46) BACE1
SCHEMBL9979870 0.62 BACE1 (0.36) BACE1NUDT1
SCHEMBL23100601 0.61 SMN1; SMN2 (0.43) BACE1NUDT1KDM4EALDH1A1
SCHEMBL23100636 0.61 BACE1 (0.63) TBXA2RBACE1NUDT1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651903-A1 BENZIMIDAZOLE RESPIRATORY SYNCYTIAL VIRUS INHIBITORS Janssen R&D Ireland (IE) 2013-10-23 EP disclosed
WO-2012080446-A1 BENZIMIDAZOLE RESPIRATORY SYNCYTIAL VIRUS INHIBITORS JANSSEN R&D IRELAND (IE) 2012-06-21 WO disclosed