SCHEMBL9942573

SCHEMBL9942573

Cc1c[nH]c2c(C)ccnc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.46
CCR5 P51681 2/20 0.46
CCR8 P51685 2/20 0.46
PSMD14 O00487 1/20 0.37
COPS5 Q92905 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
NOS3 P29474 3/20 0.35
NOS2 P35228 3/20 0.35
AR P10275 4/20 0.33
AURKA O14965 1/20 0.33
TRIM24 O15164 1/20 0.32
TRIM33 Q9UPN9 1/20 0.32
NPC1 O15118 1/20 0.31
HSP90AA1 P07900 1/20 0.31
LRRK2 Q5S007 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1984578 0.82 CCR1 (0.42) CCR1CCR5CCR8PSMD14COPS5
SCHEMBL13132297 0.77 TRIM24 (0.51) CCR1CCR5CCR8PSMD14COPS5
SCHEMBL18509077 0.77 CCR1 (0.38) CCR1CCR5CCR8PSMD14COPS5
SCHEMBL28967640 0.75 MEN1 (0.45) CCR1CCR5CCR8L3MBTL1NPC1
SCHEMBL30166973 0.75 MEN1 (0.45) CCR1CCR5CCR8L3MBTL1NPC1
SCHEMBL12238753 0.74 KDM5A (0.44) CCR1CCR5CCR8KDM5AKDM4C
SCHEMBL5329762 0.73 CCR1 (0.31) CCR1CCR5CCR8
SCHEMBL28967616 0.71 KDM5A (0.36) CCR1CCR5CCR8KDM5AKDM4C
SCHEMBL5433974 0.70
SCHEMBL12203219 0.70 CCR1 (0.65) CCR1CCR5CCR8PSMD14COPS5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363705-B1 COMPOSITION AND ANTIVIRAL ACTIVITY OF SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2012-06-13 EP disclosed