SCHEMBL9942873

SCHEMBL9942873

CN(C)C(=O)C(=O)NC12CCC(CN)(CC1)Cn1c2nc(C(=O)NCc2ccc(F)cc2)c(O)c1=O

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.50
KCNH2 Q12809 1/20 0.45
KCNE1 P15382 1/20 0.37
CCR1 P32246 1/20 0.37
KCNQ1 P51787 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ERCC1 P07992 1/20 0.35
FEN1 P39748 1/20 0.35
ERCC4 Q92889 1/20 0.35
CALCA P06881 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LIPG Q9Y5X9 1/20 0.34
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9901141 0.93 CYP2C9 (0.51) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL14212656 0.91 CYP2C9 (0.49) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL9942964 0.90 CYP2C9 (0.41) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL9901641 0.90 CYP2C9 (0.48) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL9901008 0.90 CYP2C9 (0.52) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL62449 0.90 CYP2C9 (0.52) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL9943023 0.90 CYP2C9 (0.52) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL9942967 0.89 CYP2C9 (0.48) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL9901252 0.89 CYP2C9 (0.48) CYP2C9KCNH2KCNE1CCR1KCNQ1
SCHEMBL14234672 0.87 CYP2C9 (0.53) CYP2C9KCNH2KCNE1CCR1KCNQ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078834-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed