SCHEMBL9943555

SCHEMBL9943555

CC(C)C(=O)NC(CNC(=O)OC(Cc1ccccc1)c1cncs1)CN(Cc1ccccc1)C(=O)OCc1cncs1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 20/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9943461 0.87 CYP3A4 (0.46) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL893431 0.85 CYP3A4 (0.54) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4244758 0.79 CYP3A4 (0.44) CYP3A4CYP2D6CYP2C19
SCHEMBL4252211 0.77 CYP3A4 (0.49) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL893562 0.77 CYP3A4 (0.51) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9943809 0.75 CCR6 (0.44) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL892734 0.74 CYP3A4 (0.54) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL272297 0.74 CYP3A4 (0.69) CYP3A4
SCHEMBL272296 0.74 CYP3A4 (0.69) CYP3A4
SCHEMBL4244320 0.73 CYP3A4 (0.46) CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465855-A1 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP disclosed
EP-2465856-A2 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP disclosed