SCHEMBL9943809

SCHEMBL9943809

O=C(NCCCN(Cc1ccccc1)C(=O)OCc1ccccc1)OC(Cc1ccccc1)c1cncs1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR6 P51684 1/20 0.44
PAX8 Q06710 1/20 0.44
CYP3A4 P08684 10/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
HTT P42858 1/20 0.38
REN P00797 1/20 0.35
TGM2 P21980 1/20 0.35
ANPEP P15144 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9943670 0.91 CYP3A4 (0.39) CYP3A4CYP2D6CYP2C9CYP2C19REN
SCHEMBL9943681 0.91 REN (0.39) CYP3A4CYP2D6CYP2C9CYP2C19REN
SCHEMBL9943653 0.88 HDAC3 (0.40) PAX8CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9943461 0.79 CYP3A4 (0.46) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL893112 0.75 CYP3A4 (0.57) CCR6PAX8CYP3A4CYP2D6CYP2C9
SCHEMBL9943555 0.75 CYP3A4 (0.48) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL893726 0.73 CYP3A4 (0.51) CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL893063 0.73 CYP3A4 (0.59) CCR6PAX8CYP3A4CYP2D6CYP2C9
SCHEMBL11919241 0.72 CCR6 (0.60) CCR6PAX8CYP3A4CYP2D6CYP2C9
SCHEMBL9943695 0.72 CYP3A4 (0.49) CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465856-A2 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP claimed
EP-2465855-A1 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP disclosed
EP-2465856-A2 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP disclosed