SCHEMBL9947604

SCHEMBL9947604

CC(C)Oc1c2c(c(O)c3ccccc13)C(=O)N(c1ccc(CC(=O)O)c(F)c1)C2=O

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 17/20 0.52
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 1/20 0.46
PPARG P37231 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33
FABP5 Q01469 1/20 0.33
MEN1 O00255 1/20 0.33
CYP2C9 P11712 1/20 0.33
AKR1B1 P15121 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8591107 0.95 PTGER4 (0.57) PTGER4CYP1A2CYP2D6FABP5MEN1
SCHEMBL1590674 0.91 PTGER4 (0.53) PTGER4CYP1A2CYP2D6FABP5KMT2A
SCHEMBL10058532 0.89 PTGER4 (0.45) PTGER4CYP1A2CYP2D6MEN1KMT2A
SCHEMBL9947630 0.88 PTGER4 (0.54) PTGER4CYP1A2CYP2D6MEN1KMT2A
SCHEMBL9947792 0.88 PTGER4 (0.53) PTGER4CYP1A2CYP2D6PPARGPPARD
SCHEMBL9947656 0.87 PTGER4 (0.68) PTGER4CYP1A2CYP2D6
SCHEMBL1590562 0.86 PTGER4 (0.55) PTGER4CYP1A2CYP2D6MEN1CYP2C9
SCHEMBL9948068 0.86 PTGER4 (0.58) PTGER4CYP1A2CYP2D6PPARGPPARD
SCHEMBL3967404 0.84 PTGER4 (0.68) PTGER4CYP1A2CYP2D6PPARDPPARA
SCHEMBL9606795 0.83 PTGER4 (0.48) PTGER4CYP1A2CYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979317-B1 BENZOISOINDOLE DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LTD (GB) 2012-08-22 EP disclosed
US-8207213-B2 Benzoisoindole derivatives for the treatment of pain GLAXO GROUP LIMITED (GB) 2012-06-26 US disclosed