SCHEMBL9947792

SCHEMBL9947792

O=C(O)Cc1ccc(N2C(=O)c3c(c(O)c4ccccc4c3O)C2=O)cc1F

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 9/20 0.53
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 1/20 0.43
AKR1B1 P15121 4/20 0.39
MEN1 O00255 1/20 0.39
CYP2C9 P11712 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PIM3 Q86V86 1/20 0.36
HIPK4 Q8NE63 1/20 0.36
SCN2A Q99250 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
CXCL8 P10145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9947656 0.89 PTGER4 (0.68) PTGER4CYP1A2CYP2D6
SCHEMBL14431117 0.89 PTGER4 (0.46) PTGER4CYP1A2CYP2D6AKR1B1MEN1
SCHEMBL9947604 0.88 PTGER4 (0.52) PTGER4CYP1A2CYP2D6AKR1B1MEN1
SCHEMBL9948068 0.87 PTGER4 (0.58) PTGER4CYP1A2CYP2D6PPARGPPARD
SCHEMBL10058500 0.84 PTGER4 (0.48) PTGER4CYP1A2CYP2D6MEN1KMT2A
SCHEMBL1590562 0.82 PTGER4 (0.55) PTGER4CYP1A2CYP2D6AKR1B1MEN1
SCHEMBL4611730 0.82 PTGER4 (0.74) PTGER4CYP1A2CYP2D6
SCHEMBL8591107 0.81 PTGER4 (0.57) PTGER4CYP1A2CYP2D6AKR1B1MEN1
SCHEMBL9947957 0.81 PTGER4 (0.59) PTGER4CYP1A2CYP2D6MEN1KMT2A
SCHEMBL12002249 0.81 PTGER4 (0.45) PTGER4CYP1A2CYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979317-B1 BENZOISOINDOLE DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LTD (GB) 2012-08-22 EP disclosed
US-8207213-B2 Benzoisoindole derivatives for the treatment of pain GLAXO GROUP LIMITED (GB) 2012-06-26 US disclosed