SCHEMBL9947605

SCHEMBL9947605

Cn1cnc(-c2nnc3c4cc(-c5ccccc5)c(-c5ccc(C6(NC(=O)O)CC7(C6)OCCO7)cc5)nc4ccn23)c1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 18/20 0.39
AKT2 P31751 10/20 0.39
AKT3 Q9Y243 2/20 0.39
FECH P22830 1/20 0.39
KCNH2 Q12809 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10226590 0.92 AKT1 (0.37) AKT1AKT2AKT3FECHKCNH2
SCHEMBL4286303 0.90 AKT1 (0.44) AKT1AKT2AKT3FECHKCNH2
SCHEMBL4295111 0.90 AKT1 (0.46) AKT1AKT2AKT3FECHKCNH2
SCHEMBL3627805 0.88 AKT1 (0.41) AKT1AKT2AKT3FECHKCNH2
SCHEMBL1674693 0.87 AKT1 (0.46) AKT1AKT2AKT3FECHKCNH2
SCHEMBL1674497 0.85 AKT1 (0.37) AKT1AKT2AKT3FECHKCNH2
SCHEMBL3623778 0.84 AKT1 (0.42) AKT1AKT2AKT3FECHKCNH2
SCHEMBL4289993 0.84 AKT1 (0.40) AKT1AKT2AKT3FECHKCNH2
SCHEMBL10226683 0.83 AKT1 (0.38) AKT1AKT2AKT3FECHKCNH2
SCHEMBL12583525 0.82 AKT1 (0.45) AKT1AKT2AKT3FECHKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2303269-B1 INHIBITORS OF AKT ACTIVITY MERCK SHARP & DOHME (US) 2014-07-30 EP disclosed
US-8207169-B2 Substituted [1,2,4]triazolo[4′,3′:1,6]pyrido[2,3-b]pyrazines of the formula D MSD K.K. (JP) 2012-06-26 US disclosed