SCHEMBL9952062

SCHEMBL9952062

CCOc1c(CCNc2ncnc3[nH]cnc23)cc(Cl)c(C#N)c1C1CN(CC)C1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 9/20 0.37
AXL P30530 2/20 0.35
MERTK Q12866 2/20 0.35
ALDH1A1 P00352 1/20 0.32
ABCC1 P33527 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL9953549 0.93 PIK3CD (0.35) PIK3CDAXLMERTK
SCHEMBL9953147 0.90 PIK3CD (0.37) PIK3CDAXLMERTK
Trifluoroacetic Acid SCHEMBL9952183 0.86 PIK3CD (0.37) PIK3CDAXLMERTK
SCHEMBL9929351 0.83 PIK3CD (0.44) PIK3CDAXLMERTK
SCHEMBL9960484 0.82 PIK3CD (0.35) PIK3CDALDH1A1
SCHEMBL17147215 0.79 PIK3CD (0.47) PIK3CDAXLMERTK
Trifluoroacetic Acid SCHEMBL9929573 0.78 PIK3CD (0.41) PIK3CDAXLMERTK
SCHEMBL9952900 0.78 PIK3CD (0.34) PIK3CD
SCHEMBL9952126 0.77 PDE5A (0.33)
SCHEMBL9929054 0.76 PIK3CD (0.43) PIK3CDAXLMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655374-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS Incyte Corporation (US) 2013-10-30 EP claimed
WO-2012087881-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2012-06-28 WO claimed
EP-2655374-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS Incyte Corporation (US) 2013-10-30 EP disclosed
WO-2012087881-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2012-06-28 WO disclosed