SCHEMBL9953600

SCHEMBL9953600

CN(C)c1ncc(-c2ccc3nc(N)n(-c4ccccc4)c(=O)c3c2)cn1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 13/20 0.57
PIK3CG P48736 10/20 0.57
ALDH1A1 P00352 6/20 0.47
CYP1A2 P05177 6/20 0.47
CASP1 P29466 6/20 0.47
CASP7 P55210 6/20 0.47
MEN1 O00255 5/20 0.47
USP2 O75604 5/20 0.47
KMT2A Q03164 5/20 0.47
HIF1A Q16665 3/20 0.47
CYP3A4 P08684 1/20 0.47
HSD17B10 Q99714 4/20 0.46
CYP2D6 P10635 2/20 0.46
ALOX15 P16050 2/20 0.46
TSHR P16473 1/20 0.46
LMNA P02545 1/20 0.46
BRCA1 P38398 1/20 0.44
HBB P68871 1/20 0.44
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953490 0.84 PI4KA (0.65) PI4KAPIK3CGALDH1A1CYP1A2CASP1
SCHEMBL9953522 0.81 PI4KA (0.73) PI4KAPIK3CGCASP1
SCHEMBL10288670 0.81 PI4KA (0.57) PI4KAPIK3CGALDH1A1LMNA
SCHEMBL10288673 0.80 PI4KA (0.56) PI4KAPIK3CGCYP3A4
SCHEMBL9955010 0.80 PI4KA (0.59) PI4KAPIK3CGALDH1A1LMNA
SCHEMBL9954494 0.80 PI4KA (0.63) PI4KAPIK3CG
SCHEMBL9954698 0.78 PI4KA (0.72) PI4KAPIK3CG
SCHEMBL9953082 0.78 PI4KA (0.70) PI4KAPIK3CG
SCHEMBL10288761 0.77 PI4KA (0.57) PI4KAPIK3CGALDH1A1LMNA
SCHEMBL9954452 0.77 PI4KA (0.69) PI4KAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed