SCHEMBL9955412

SCHEMBL9955412

Cc1ncoc1-c1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.47
MAPK14 Q16539 1/20 0.44
IMPDH2 P12268 1/20 0.44
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
ACHE P22303 1/20 0.39
PIM1 P11309 1/20 0.38
CYP17A1 P05093 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
HCRTR2 O43614 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
ESR2 Q92731 1/20 0.38
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9956334 0.82 IMPDH2 (0.56) NOTUMMAPK14IMPDH2ACHEHCRTR2
SCHEMBL9956542 0.79 NOTUM (0.47) NOTUMMAPK14KDM4EMAPTCYP17A1
SCHEMBL3441822 0.79 MAP4K4 (0.47) IMPDH2KDM4EMAPTSMN1; SMN2
SCHEMBL27422553 0.79 IMPDH2 (0.47) IMPDH2ACHECYP3A4
SCHEMBL9953638 0.79 NOTUM (0.47) NOTUMMAPK14IMPDH2MAPTHCRTR2
SCHEMBL472496 0.79 IMPDH2 (0.41) MAPK14IMPDH2
SCHEMBL1855319 0.79 NOTUM (0.51) NOTUMIMPDH2KDM4ECYP3A4GAA
SCHEMBL472455 0.78 MAPK14 (0.54) NOTUMMAPK14IMPDH2
SCHEMBL343219 0.77 ADORA2A (0.50) NOTUMMAPK14IMPDH2KDM4EMAPT
SCHEMBL9954145 0.76 NOTUM (0.44) NOTUMMAPK14KDM4EMAPTCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed