SCHEMBL9955679

SCHEMBL9955679

C(=Cc1ccc2c(c1)OCO2)CCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.55
ATM Q13315 1/20 0.55
MAOB P27338 5/20 0.55
TRPM8 Q7Z2W7 4/20 0.51
MAOA P21397 3/20 0.51
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
CYP19A1 P11511 2/20 0.49
KMT2A Q03164 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
RAB9A P51151 2/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9955675 1.00 CYP3A4 (0.55) CYP3A4ATMMAOBTRPM8MAOA
SCHEMBL16052903 0.85 CYP3A4 (0.54) CYP3A4ATMMAOBTRPM8MAOA
SCHEMBL16052904 0.85 CYP3A4 (0.54) CYP3A4ATMMAOBTRPM8MAOA
SCHEMBL11011121 0.78 CYP3A4 (0.62) CYP3A4ATMTRPM8MAOAHDAC3
SCHEMBL8606599 0.78 ALDH1A1 (0.56) CYP3A4ATMMAOBTRPM8MAOA
SCHEMBL11011119 0.78 CYP3A4 (0.62) CYP3A4ATMTRPM8MAOAHDAC3
SCHEMBL19097963 0.77 CYP19A1 (0.71) CYP3A4ATMMAOBTRPM8CYP19A1
SCHEMBL1666984 0.77 CYP19A1 (0.71) CYP3A4ATMMAOBTRPM8CYP19A1
SCHEMBL11815830 0.75 MAOB (0.56) CYP3A4ATMMAOBTRPM8MAOA
SCHEMBL11815824 0.75 MAOB (0.56) CYP3A4ATMMAOBTRPM8MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655307-B1 COMPOUNDS CAPABLE OF RELEASING FRAGRANT COMPOUNDS GIVAUDAN SA (CH) 2018-08-01 EP claimed
EP-2655307-A1 COMPOUNDS CAPABLE OF RELEASING FRAGRANT COMPOUNDS Givaudan SA (CH) 2013-10-30 EP claimed
WO-2012085287-A1 COMPOUNDS CAPABLE OF RELEASING FRAGRANT COMPOUNDS GIVAUDAN SA (CH) 2012-06-28 WO claimed
EP-2655307-A1 COMPOUNDS CAPABLE OF RELEASING FRAGRANT COMPOUNDS Givaudan SA (CH) 2013-10-30 EP disclosed
WO-2012085287-A1 COMPOUNDS CAPABLE OF RELEASING FRAGRANT COMPOUNDS GIVAUDAN SA (CH) 2012-06-28 WO disclosed