SCHEMBL9956489

SCHEMBL9956489

Cc1ccc(-n2nccn2)c(C(=O)N2CCC3CN(C(=O)OC(C)(C)C)C3C2)c1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 18/20 0.64
HCRTR2 O43614 18/20 0.64
SPR P35270 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9957752 0.93 HCRTR2 (0.59) HCRTR1HCRTR2SPR
SCHEMBL9954161 0.88 SPR (0.51) HCRTR1HCRTR2SPR
SCHEMBL9954160 0.88 SPR (0.51) HCRTR1HCRTR2SPR
SCHEMBL9955001 0.86 HCRTR2 (0.71) HCRTR1HCRTR2
SCHEMBL30670421 0.84 HCRTR1 (0.61) HCRTR1HCRTR2
SCHEMBL3102096 0.83 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL9957016 0.82 HCRTR2 (0.65) HCRTR1HCRTR2
SCHEMBL17859340 0.82 HCRTR1 (0.66) HCRTR1HCRTR2
SCHEMBL19549869 0.82 HCRTR1 (0.66) HCRTR1HCRTR2
SCHEMBL19549868 0.82 HCRTR1 (0.66) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed