SCHEMBL9957634

SCHEMBL9957634

Cc1ccc(-n2nccn2)c(C(=O)N2CC3CCN(c4nc5cc(F)ccc5o4)C[C@H]32)c1F

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 20/20 0.56
HCRTR1 O43613 19/20 0.56
NR1I2 O75469 1/20 0.46
ADRA2B P18089 1/20 0.46
KCNH2 Q12809 1/20 0.46
CYP3A4 P08684 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954737 0.84 HCRTR1 (0.69) HCRTR2HCRTR1
SCHEMBL9956544 0.84 HCRTR1 (0.57) HCRTR2HCRTR1
SCHEMBL9957554 0.84 HCRTR1 (0.57) HCRTR2HCRTR1
SCHEMBL9957552 0.84 HCRTR1 (0.57) HCRTR2HCRTR1
SCHEMBL9957079 0.84 HCRTR1 (0.57) HCRTR2HCRTR1
SCHEMBL9957650 0.81 HCRTR1 (0.56) HCRTR2HCRTR1
SCHEMBL9957647 0.81 HCRTR1 (0.56) HCRTR2HCRTR1
SCHEMBL9957712 0.76 HCRTR1 (0.49) HCRTR2HCRTR1CYP3A4
SCHEMBL9957873 0.75 HCRTR1 (0.51) HCRTR2HCRTR1
SCHEMBL9956269 0.74 HCRTR1 (0.66) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed