SCHEMBL9958718

SCHEMBL9958718

NS(=O)(=O)c1cccc(-c2cccc(-c3nc(-c4ccc(F)cc4)cc(C(F)(F)F)n3)n2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.50
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
STAT3 P40763 2/20 0.50
STAT1 P42224 2/20 0.50
RAB9A P51151 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
TLR9 Q9NR96 2/20 0.50
MITF O75030 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
PTGS2 P35354 5/20 0.43
TP53 P04637 2/20 0.43
MAPK1 P28482 2/20 0.43
HSD17B10 Q99714 2/20 0.43
SDHB P21912 2/20 0.43
SYK P43405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3567232 0.91 KIF11 (0.45) KDM4ELMNASTAT3STAT1RAB9A
SCHEMBL3569106 0.90 KDM4E (0.53) KDM4EALDH1A1LMNASTAT3STAT1
SCHEMBL3568481 0.86 SYK (0.47) KDM4EALDH1A1LMNASTAT3STAT1
SCHEMBL3564767 0.81
SCHEMBL3568722 0.80 PTGES2 (0.48) LMNASTAT3STAT1RAB9ANPSR1
SCHEMBL3564758 0.80 LRRK2 (0.43) MAOAMAOBCA2CA9PTGS2
SCHEMBL3560858 0.79 KDM4E (0.53) KDM4EALDH1A1MAOBCA2CA9
SCHEMBL3568564 0.79 KDM4E (0.47) KDM4EALDH1A1LMNASTAT3STAT1
SCHEMBL3564023 0.79 KIF11 (0.56) PTGS2PTGS1
SCHEMBL2402375 0.78 LRRK2 (0.47) PTGS2SYKPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468727-A1 Pyridine and pyrimidine derivatives as MGLUR2 antagonists F. Hoffmann-La Roche AG (CH) 2012-06-27 EP claimed