SCHEMBL9959352

SCHEMBL9959352

CCCCCCC=CC[SiH](C)Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 5/20 0.50
TRPV1 Q8NER1 1/20 0.50
TERT O14746 3/20 0.44
PTPN1 P18031 3/20 0.44
PPARG P37231 3/20 0.44
PPARD Q03181 3/20 0.44
PPARA Q07869 3/20 0.44
CYP1A2 P05177 2/20 0.44
MAPT P10636 2/20 0.44
CYP2C19 P33261 2/20 0.44
BLM P54132 2/20 0.44
HSD17B10 Q99714 2/20 0.44
FABP4 P15090 2/20 0.44
KMT2A Q03164 2/20 0.44
GMNN O75496 1/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5572876 0.91 FAAH (0.38) FAAHTRPV1PPARACYP1A2MAPT
SCHEMBL6248715 0.84 FAAH (0.52) FAAHTRPV1TERTPTPN1PPARG
SCHEMBL4355517 0.84 FAAH (0.52) FAAHTRPV1TERTPTPN1PPARG
SCHEMBL4357218 0.84 FAAH (0.52) FAAHTRPV1TERTPTPN1PPARG
SCHEMBL4349965 0.82 FAAH (0.48) FAAHTRPV1TERTPTPN1PPARG
SCHEMBL25362976 0.78 FAAH (0.74) FAAHTRPV1TERTPTPN1PPARG
SCHEMBL23291808 0.78 FAAH (0.74) FAAHTRPV1TERTPTPN1PPARG
SCHEMBL21366450 0.78 FAAH (0.74) FAAHTRPV1TERTPTPN1PPARG
SCHEMBL24218814 0.78 FAAH (0.74) FAAHTRPV1TERTPTPN1PPARG
SCHEMBL22654062 0.78 FAAH (0.74) FAAHTRPV1TERTPTPN1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697266-B1 METHOD FOR PREPARING A MASTERBATCH OF AN ELASTOMER AND AN INORGANIC REINFORCING FILLER MICHELIN & CIE (FR) 2017-02-22 EP claimed
EP-2655422-B1 PROCESS FOR PREPARING A MASTERBATCH IN THE LIQUID PHASE MICHELIN & CIE (FR) 2015-02-25 EP claimed
EP-2697266-A1 METHOD FOR PREPARING A MASTERBATCH OF AN ELASTOMER AND AN INORGANIC REINFORCING FILLER Compagnie Générale des Etablissements Michelin (FR) 2014-02-19 EP claimed
EP-2655422-A1 PROCESS FOR PREPARING A MASTERBATCH IN THE LIQUID PHASE Compagnie Générale des Etablissements Michelin (FR) 2013-10-30 EP claimed
WO-2012139669-A1 METHOD FOR PREPARING A MASTERBATCH OF AN ELASTOMER AND AN INORGANIC REINFORCING FILLER COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2012-10-18 WO claimed
WO-2012085137-A1 PROCESS FOR PREPARING A MASTERBATCH IN THE LIQUID PHASE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2012-06-28 WO claimed
EP-2697266-B1 METHOD FOR PREPARING A MASTERBATCH OF AN ELASTOMER AND AN INORGANIC REINFORCING FILLER MICHELIN & CIE (FR) 2017-02-22 EP disclosed
EP-2655423-B1 PROCESS FOR PREPARING A MASTERBATCH IN THE LIQUID PHASE MICHELIN & CIE (FR) 2015-03-25 EP disclosed
EP-2655422-B1 PROCESS FOR PREPARING A MASTERBATCH IN THE LIQUID PHASE MICHELIN & CIE (FR) 2015-02-25 EP disclosed
EP-2697266-A1 METHOD FOR PREPARING A MASTERBATCH OF AN ELASTOMER AND AN INORGANIC REINFORCING FILLER Compagnie Générale des Etablissements Michelin (FR) 2014-02-19 EP disclosed
EP-2655423-A1 PROCESS FOR PREPARING A MASTERBATCH IN THE LIQUID PHASE Compagnie Générale des Etablissements Michelin (FR) 2013-10-30 EP disclosed
WO-2012139669-A1 METHOD FOR PREPARING A MASTERBATCH OF AN ELASTOMER AND AN INORGANIC REINFORCING FILLER COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2012-10-18 WO disclosed
WO-2012085135-A1 PROCESS FOR PREPARING A MASTERBATCH IN THE LIQUID PHASE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2012-06-28 WO disclosed