SCHEMBL9959918

SCHEMBL9959918

Fc1ccc(Nc2ncc3c(n2)CCCC3)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 9/20 0.74
CDK5R1 Q15078 9/20 0.74
CCNA2 P20248 7/20 0.74
CDK2 P24941 7/20 0.74
GRM5 P41594 5/20 0.74
CDK1 P06493 2/20 0.59
CCNB1 P14635 2/20 0.59
MAOB P27338 2/20 0.59
CCNT1 O60563 1/20 0.53
CCNE1 P24864 1/20 0.53
CCND3 P30281 1/20 0.53
FLT3 P36888 1/20 0.53
CDK9 P50750 1/20 0.53
CDK6 Q00534 1/20 0.53
AURKA O14965 1/20 0.53
GRM1 Q13255 1/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9959938 0.85 GRM5 (1.00) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL9959836 0.84 CDK5 (1.00) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL23656974 0.80 GRM5 (0.72) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL9959309 0.80 CDK5 (0.49) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL23020744 0.78 AURKA (0.51) CDK5CDK5R1CCNA2CDK2GRM5
Hydrochloric Acid SCHEMBL23000039 0.77 AURKA (0.50) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL11299433 0.75 IKBKB (0.71) CDK5CDK5R1CCNA2CDK2AURKA
SCHEMBL9960032 0.74 GRM5 (1.00) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL12498045 0.74 MAPK1 (0.58) CDK5CDK5R1CDK2MAPTMAPK1
SCHEMBL12609744 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085166-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO claimed
WO-2012085166-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO disclosed