SCHEMBL9959938

SCHEMBL9959938

Clc1ccc(Nc2ncc3c(n2)CCCC3)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 1.00
CDK5 Q00535 9/20 0.74
CDK5R1 Q15078 9/20 0.74
CCNA2 P20248 9/20 0.74
CDK2 P24941 9/20 0.74
MAOB P27338 3/20 0.71
MAOA P21397 2/20 0.63
CDK1 P06493 2/20 0.59
CCNB1 P14635 2/20 0.59
CCNT1 O60563 1/20 0.53
CCNE1 P24864 1/20 0.53
CCND3 P30281 1/20 0.53
FLT3 P36888 1/20 0.53
CDK9 P50750 1/20 0.53
CDK6 Q00534 1/20 0.53
MAPT P10636 1/20 0.48
EGFR P00533 1/20 0.48
KDR P35968 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9959918 0.85 CDK5 (0.74) GRM5CDK5CDK5R1CCNA2CDK2
SCHEMBL9959836 0.84 CDK5 (1.00) GRM5CDK5CDK5R1CCNA2CDK2
SCHEMBL9960032 0.83 GRM5 (1.00) GRM5CDK5CDK5R1CCNA2CDK2
SCHEMBL23656973 0.80 GRM5 (0.95) GRM5CCNA2CDK2MAOBMAOA
SCHEMBL9955104 0.77 GRM5 (1.00) GRM5CCNA2CDK2MAOBMAOA
Hydrochloric Acid SCHEMBL22999918 0.77 GRM5 (0.62) GRM5CDK5CDK5R1CCNA2CDK2
SCHEMBL11296762 0.75 IKBKB (0.71) GRM5CDK5CDK5R1CCNA2CDK2
SCHEMBL12609744 0.73
SCHEMBL12609743 0.73
SCHEMBL1594953 0.72 CDK5 (0.58) GRM5CDK5CDK5R1CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085166-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO claimed
WO-2012085166-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO disclosed