SCHEMBL9959960

SCHEMBL9959960

COCNC(=O)C1CCc2nc(Nc3cccc(Cl)c3)ncc2C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.53
MAOB P27338 2/20 0.53
MAOA P21397 1/20 0.46
CNR2 P34972 11/20 0.45
CDK5 Q00535 3/20 0.44
CDK5R1 Q15078 3/20 0.44
CCNA2 P20248 2/20 0.44
CDK2 P24941 2/20 0.44
CYP3A4 P08684 4/20 0.43
CYP2C9 P11712 4/20 0.43
CYP2C19 P33261 4/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
ALK Q9UM73 1/20 0.42
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954113 0.85 GRM5 (0.61) GRM5MAOBMAOACNR2CDK5
SCHEMBL9954136 0.84 GRM5 (0.54) GRM5MAOBMAOACNR2CDK5
SCHEMBL9956217 0.83 GRM5 (0.57) GRM5MAOBMAOACNR2CDK5
SCHEMBL9954096 0.80 GRM5 (0.58) GRM5MAOBMAOACNR2CDK5
SCHEMBL9956051 0.75 GRM5 (0.59) GRM5MAOBMAOACNR2CDK5
SCHEMBL9954695 0.72 PDGFRB (0.66) GRM5MAOBMAOAKDR
SCHEMBL9955388 0.72 GRM5 (0.58) GRM5MAOBMAOAKDR
SCHEMBL9954811 0.71 GRM5 (0.59) GRM5MAOBMAOACNR2CYP3A4
SCHEMBL9960032 0.71 GRM5 (1.00) GRM5MAOBMAOACDK5CDK5R1
SCHEMBL9955865 0.70 PDGFRB (0.55) GRM5MAOBMAOAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085167-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-06-28 WO disclosed