SCHEMBL9965131

SCHEMBL9965131

Nc1cccc(C(C(c2cccnc2)c2cccnc2)n2ccnn2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.41
MEN1 O00255 1/20 0.41
PSIP1 O75475 1/20 0.41
AXL P30530 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TEK Q02763 1/20 0.35
CFTR P13569 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
GOPC Q9HD26 1/20 0.34
CYP17A1 P05093 1/20 0.34
KCNA5 P22460 5/20 0.34
KCND3 Q9UK17 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CYP11B1 P15538 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1243818 0.87 CYP19A1 (0.49) CYP19A1SMN1; SMN2CFTRSLC6A2SLC6A4
SCHEMBL9965186 0.86 CYP19A1 (0.43) CYP19A1MEN1PSIP1AXLMKNK1
SCHEMBL9965132 0.86 KCNA5 (0.40) CYP19A1MEN1PSIP1AXLMKNK1
SCHEMBL1242145 0.83 CYP19A1 (0.45) CYP19A1CYP17A1KCNA5CYP11B1
SCHEMBL1242629 0.77 CYP19A1 (0.57) CYP19A1CYP17A1KCNA5CYP11B1
SCHEMBL1243320 0.76 CYP19A1 (0.44) CYP19A1SMN1; SMN2CFTRSLC6A2SLC6A4
SCHEMBL17064640 0.74 SMN1; SMN2 (0.65) CYP19A1MEN1PSIP1AXLMKNK1
SCHEMBL12890821 0.71 KCNA5 (0.36) CYP19A1KCNA5
SCHEMBL1242323 0.71 CYP19A1 (0.39) CYP19A1KCNA5KDM4E
SCHEMBL1242375 0.70 CFTR (0.41) CYP19A1SMN1; SMN2CFTRSLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082746-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-06-21 WO disclosed