SCHEMBL9965157

SCHEMBL9965157

CC(C)C(c1ccc2cc(N)ccc2c1)n1ccnn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 4/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
CYP19A1 P11511 4/20 0.39
NOTUM Q6P988 1/20 0.36
ALDH1A1 P00352 5/20 0.33
CYP3A4 P08684 2/20 0.33
HSD17B10 Q99714 2/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
LMNA P02545 2/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
HBB P68871 1/20 0.33
HIF1A Q16665 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
F2 P00734 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9945351 0.86 CYP17A1 (0.46) CYP17A1CYP2C9CYP2C19CYP19A1NOTUM
SCHEMBL9895460 0.83 CYP2C9 (0.50) CYP17A1CYP2C9CYP2C19NOTUMLMNA
SCHEMBL9896985 0.82 CYP17A1 (0.53) CYP17A1CYP2C9CYP2C19CYP19A1CYP3A4
SCHEMBL9895663 0.82 CYP17A1 (0.65) CYP17A1CYP2C9CYP2C19CYP19A1NOTUM
SCHEMBL9895228 0.81 CYP19A1 (0.55) CYP17A1CYP2C9CYP2C19CYP19A1CYP3A4
SCHEMBL9896161 0.80 CYP17A1 (0.67) CYP17A1CYP2C9CYP2C19CYP19A1CYP3A4
SCHEMBL9894973 0.80 CYP17A1 (0.50) CYP17A1CYP2C9CYP2C19CYP19A1CYP3A4
SCHEMBL9965128 0.80 KDM4E (0.42) CYP19A1ALDH1A1HSD17B10MEN1KMT2A
SCHEMBL9945352 0.79 CYP2C19 (0.49) CYP17A1CYP2C9CYP2C19CYP19A1ALDH1A1
SCHEMBL9895951 0.79 CYP17A1 (0.53) CYP17A1CYP2C9CYP2C19CYP19A1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082746-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-06-21 WO disclosed