SCHEMBL9965128

SCHEMBL9965128

CC(C)C(c1ccc2cc(N)ccc2n1)n1ccnn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
POLB P06746 2/20 0.42
CASP6 P55212 1/20 0.42
PLAU P00749 1/20 0.41
HTT P42858 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
F2 P00734 1/20 0.37
CHRM2 P08172 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
MAOA P21397 1/20 0.37
DRD1 P21728 1/20 0.37
ACHE P22303 1/20 0.37
PTGS1 P23219 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
OPRM1 P35372 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9895726 0.84 NCF1 (0.46) KDM4ELMNAPOLBMEN1KMT2A
SCHEMBL9896964 0.83 AAK1 (0.44) MAOAKCNH2AAK1ATMCYP19A1
SCHEMBL9894903 0.83 CYP19A1 (0.45) KCNH2HRH3AAK1CYP19A1
SCHEMBL9894682 0.82 CYP19A1 (0.42) AAK1CYP19A1
SCHEMBL9894758 0.82 CYP19A1 (0.36) AAK1CYP19A1
SCHEMBL9896553 0.81 CYP17A1 (0.50) AAK1
SCHEMBL9945353 0.81 NCF1 (0.39) KDM4ELMNAHTTMEN1KMT2A
SCHEMBL9896550 0.80 MAOA (0.38) LMNAADORA3MAOASLC6A2SLC6A3
SCHEMBL9965157 0.80 CYP17A1 (0.43) KDM4ELMNAPOLBCASP6PLAU
SCHEMBL9895652 0.77 CYP17A1 (0.53) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082746-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-06-21 WO disclosed