SCHEMBL9965460

SCHEMBL9965460

CC(C)CC(=O)N1CCC(C(=O)Nc2ccccc2Oc2ccc(CC(F)(F)F)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.50
TRPV1 Q8NER1 3/20 0.50
PTPN1 P18031 1/20 0.49
GAA P10253 1/20 0.49
PKM P14618 1/20 0.49
KMT2A Q03164 1/20 0.47
ACHE P22303 1/20 0.45
BACE1 P56817 1/20 0.45
NAMPT P43490 1/20 0.44
ALDH1A1 P00352 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MGLL Q99685 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965373 0.89 EPHX2 (0.52) POLBTRPV1PTPN1GAAPKM
SCHEMBL9965405 0.89 GAA (0.51) POLBTRPV1PTPN1GAAPKM
SCHEMBL10173900 0.81 PTPN1 (0.53) POLBTRPV1PTPN1GAAPKM
SCHEMBL14639696 0.80 PTPN1 (0.49) POLBTRPV1PTPN1GAAPKM
SCHEMBL14639656 0.79 PTPN1 (0.49) POLBTRPV1PTPN1GAAPKM
SCHEMBL9965372 0.78 GAA (0.55) POLBTRPV1GAAPKMKMT2A
SCHEMBL9965424 0.77 GAA (0.52) POLBGAAPKMKMT2AACHE
SCHEMBL9965371 0.77 EPHX2 (0.55) POLBTRPV1GAAPKMKMT2A
SCHEMBL9965382 0.76 PTPN1 (0.51) POLBTRPV1PTPN1GAAPKM
SCHEMBL14639655 0.75 GAA (0.52) POLBTRPV1GAAPKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-B1 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS STERIX LTD (GB) 2012-06-20 EP disclosed