SCHEMBL14639655

SCHEMBL14639655

CC(C)OC(=O)N1CCC(C(=O)Nc2ccccc2Oc2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.52
PKM P14618 1/20 0.52
KMT2A Q03164 1/20 0.49
ACHE P22303 1/20 0.47
BACE1 P56817 1/20 0.47
TRPV1 Q8NER1 1/20 0.46
SCN1A P35498 1/20 0.44
SCN5A Q14524 1/20 0.44
SCN9A Q15858 1/20 0.44
ALDH1A1 P00352 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
POLB P06746 2/20 0.43
UBE2M P61081 1/20 0.43
DCUN1D1 Q96GG9 1/20 0.43
MGLL Q99685 1/20 0.43
MMP1 P03956 1/20 0.42
MMP13 P45452 1/20 0.42
LIPE Q05469 1/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965372 0.89 GAA (0.55) GAAPKMKMT2AACHEBACE1
SCHEMBL642298 0.89 GAA (0.54) GAAPKMKMT2AACHEBACE1
SCHEMBL9965416 0.87 GAA (0.57) GAAPKMKMT2AACHEBACE1
SCHEMBL9965373 0.86 EPHX2 (0.52) GAAPKMKMT2AACHEBACE1
SCHEMBL9965380 0.83 GAA (0.55) GAAPKMKMT2AACHEBACE1
SCHEMBL9965370 0.83 ACHE (0.66) GAAPKMKMT2AACHEBACE1
SCHEMBL9965384 0.83 GAA (0.54) GAAPKMKMT2AACHEBACE1
SCHEMBL9965371 0.81 EPHX2 (0.55) GAAPKMKMT2AACHEBACE1
SCHEMBL641560 0.79 GAA (0.54) GAAPKMKMT2AACHEBACE1
SCHEMBL640944 0.79 GAA (0.62) GAAPKMKMT2ARXFP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007003934-A2 17BETA-HYDR0XYSTER0ID DEHYDROGENASE TYPE 3 (17BETA-HSD3 ) INHIBITORS STERIX LIMITED (GB) 2007-01-11 WO disclosed