SCHEMBL9967201

SCHEMBL9967201

Cc1ccnc(-c2c[nH]c3ncc(F)cc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 9/20 0.47
CCNA2 P20248 9/20 0.47
CDK2 P24941 9/20 0.47
CDK9 P50750 9/20 0.47
LRRK2 Q5S007 1/20 0.44
CCR1 P32246 1/20 0.43
CCR5 P51681 1/20 0.43
CCR8 P51685 1/20 0.43
CCNB2 O95067 1/20 0.41
CDK1 P06493 1/20 0.41
RET P07949 1/20 0.41
CCNB1 P14635 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
KIT P10721 2/20 0.40
METAP2 P50579 1/20 0.40
CLK1 P49759 1/20 0.40
CLK2 P49760 1/20 0.40
DYRK1A Q13627 1/20 0.40
DYRK2 Q92630 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9967203 0.79 GSK3A (0.43) CCNT1CCNA2CDK2CDK9KIT
SCHEMBL1836259 0.77 CCNT1 (0.76) CCNT1CCNA2CDK2CDK9PDPK1
SCHEMBL20846122 0.74 KIT (0.51) CDK2CDK1KITCLK1CLK2
SCHEMBL23655695 0.73 CDK2 (0.45) CCNT1CCNA2CDK2CDK9CLK1
SCHEMBL26174709 0.73 PRKCI (0.54) CCNT1CCNA2CDK2CDK9LRRK2
SCHEMBL24059791 0.72 GSK3A (0.48) CDK2CLK1CLK2DYRK1ADYRK2
SCHEMBL15345020 0.72 CCR1 (0.43) CCR1CCR5CCR8CCNB2CDK1
SCHEMBL14041214 0.72 MET (0.43) KIT
SCHEMBL15345166 0.71 MET (0.48) CCNT1CCNA2CDK2CDK9CCR1
SCHEMBL20561743 0.71 KIT (0.39) CDK2KITCLK1CLK2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083122-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICAL INCORPORATED (US) 2012-06-21 WO disclosed