SCHEMBL9967225

SCHEMBL9967225

N#Cc1cc(F)c(N)nc1-c1c[nH]c2ncc(Cl)cc12

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KHK P50053 1/20 0.46
JAK2 O60674 1/20 0.44
CHUK O15111 2/20 0.37
CCNT1 O60563 2/20 0.36
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
CDK9 P50750 2/20 0.36
MAP3K14 Q99558 1/20 0.36
NTRK1 P04629 2/20 0.36
PIK3CA P42336 1/20 0.36
KIT P10721 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9967124 0.88 KHK (0.42) KHKJAK2CHUKCCNT1CCNA2
SCHEMBL22883822 0.84 RPS6KA5 (0.46) KHKCHUKCCNT1CDK2CDK9
SCHEMBL9967446 0.82 MAP3K14 (0.48) JAK2CHUKCCNT1CCNA2CDK2
SCHEMBL17518539 0.81 KHK (0.48) KHKCHUKMAP3K14
SCHEMBL8943059 0.76 JAK2 (0.50) JAK2
SCHEMBL18306309 0.76 JAK2 (0.53) JAK2CCNT1CCNA2CDK2CDK9
SCHEMBL22963816 0.74 GSK3A (0.39) JAK2CCNT1CDK2CDK9PIK3CA
SCHEMBL17518094 0.74 KHK (0.43) KHKCHUK
SCHEMBL19124511 0.73 JAK2 (0.35) JAK2
SCHEMBL9967235 0.73 CDK2 (0.42) JAK2CCNT1CCNA2CDK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083122-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICAL INCORPORATED (US) 2012-06-21 WO disclosed