SCHEMBL9967446

SCHEMBL9967446

N#Cc1cnc(N)nc1-c1c[nH]c2ncc(Cl)cc12

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 2/20 0.48
JAK2 O60674 1/20 0.47
CCNT1 O60563 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CDK9 P50750 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAP3K11 Q16584 1/20 0.41
CLK1 P49759 5/20 0.39
CDK5 Q00535 4/20 0.39
CDK5R1 Q15078 4/20 0.39
CHUK O15111 3/20 0.39
NTRK1 P04629 2/20 0.38
PIK3CA P42336 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15722386 0.85 ADORA2A (0.43) MAP3K14CCNT1CCNA2CDK2CDK9
SCHEMBL9967129 0.82 CCNT1 (0.46) CCNT1CCNA2CDK2CDK9ADORA2A
SCHEMBL9967225 0.82 KHK (0.46) MAP3K14JAK2CCNT1CCNA2CDK2
SCHEMBL1613323 0.75 CLK1 (0.69) MAP3K14ADORA2AADORA1CLK1CDK5
SCHEMBL11989895 0.74 CDK1 (0.39) JAK2CDK2CYP3A4CDK5CDK5R1
SCHEMBL14712228 0.73 JAK2 (0.52) MAP3K14JAK2CCNT1CCNA2CDK2
SCHEMBL28674867 0.71 PDPK1 (0.52) MAP3K14JAK2CCNT1CCNA2CDK2
SCHEMBL30301157 0.71 PDPK1 (0.52) MAP3K14JAK2CCNT1CCNA2CDK2
SCHEMBL14147113 0.71 HSP90AB1 (0.37) JAK2CDK2MAP3K11CLK1CDK5
SCHEMBL8941597 0.70 JAK2 (0.68) JAK2CDK2MAP3K11CLK1CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083122-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICAL INCORPORATED (US) 2012-06-21 WO disclosed