SCHEMBL997018

SCHEMBL997018

N[C@@](C=O)(c1ccc(F)cc1)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(Cl)cc2)C1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.64
CYP3A4 P08684 1/20 0.42
PTGDR2 Q9Y5Y4 2/20 0.37
TP53 P04637 2/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 2/20 0.33
P2RX7 Q99572 1/20 0.33
ALOX5 P09917 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2068537 0.78 KCNH2 (1.00) KCNH2CYP3A4PTGDR2P2RX7
SCHEMBL1052384 0.76 KCNH2 (0.82) KCNH2CYP3A4PTGDR2MAPTP2RX7
SCHEMBL2067454 0.76 KCNH2 (0.82) KCNH2CYP3A4PTGDR2MAPTP2RX7
SCHEMBL2067365 0.74 KCNH2 (0.77) KCNH2CYP3A4TP53GAAMAPT
SCHEMBL2069967 0.74 KCNH2 (0.74) KCNH2CYP3A4PTGDR2MAPTP2RX7
SCHEMBL2068572 0.74 KCNH2 (0.76) KCNH2CYP3A4PTGDR2P2RX7
SCHEMBL12952195 0.74 KCNH2 (0.74) KCNH2CYP3A4PTGDR2MAPTP2RX7
SCHEMBL20121561 0.73 KCNH2 (0.76) KCNH2CYP3A4PTGDR2P2RX7
SCHEMBL20121606 0.73 KCNH2 (0.68) KCNH2CYP3A4PTGDR2MAPTP2RX7
SCHEMBL997017 0.73 KCNH2 (0.70) KCNH2CYP3A4PTGDR2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451814-A2 FUSED IMIDAZOLES AND COMPOSITIONS COMPRISING THEM FOR THE TREATMENT OF PARASITIC DISEASES, SUCH AS E.G. MALARIA IRM LLC (BM) 2012-05-16 EP claimed
WO-2011006143-A2 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES IRM LLC (BM) 2011-01-13 WO claimed