SCHEMBL9971366

SCHEMBL9971366

COC1O[C@H](COS(=O)(=O)c2ccc(C)cc2)[C@@H](O)[C@H](O)[C@H]1NC(=O)/C=C/c1ccc(Cl)c(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HK1 P19367 2/20 0.62
HK2 P52789 2/20 0.62
CA2 P00918 5/20 0.51
CA9 Q16790 5/20 0.51
CA1 P00915 1/20 0.42
ALDH1A1 P00352 1/20 0.39
PTGS2 P35354 1/20 0.39
NOS3 P29474 2/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
PYGL P06737 4/20 0.38
MMP9 P14780 1/20 0.36
MMP12 P39900 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9937895 0.83 HK1 (0.76) HK1HK2CA2CA9CA1
SCHEMBL9937889 0.83 HK1 (0.76) HK1HK2CA2CA9CA1
SCHEMBL9938828 0.82 HK1 (0.63) HK1HK2CA2CA9NOS3
SCHEMBL9938825 0.82 HK1 (0.63) HK1HK2CA2CA9NOS3
SCHEMBL24256704 0.81 CA2 (0.53) CA2CA9CA1ALDH1A1MMP9
SCHEMBL7150215 0.81 CA2 (0.53) CA2CA9CA1ALDH1A1MMP9
SCHEMBL7150922 0.81 CA2 (0.53) CA2CA9CA1ALDH1A1MMP9
SCHEMBL16025453 0.78 CA9 (0.71) HK1HK2CA2CA9CA1
SCHEMBL16011459 0.77 CA2 (0.82) HK1HK2CA2CA9CA1
SCHEMBL16011460 0.77 CA2 (0.82) HK1HK2CA2CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083145-A1 GLUCOSAMINE DERIVATIVES GLAXO WELLCOME MANUFACTURING PTE LTD (SG) 2012-06-21 WO disclosed