SCHEMBL997226

SCHEMBL997226

COc1ccc(/C=C/C(=O)c2cc3c(cc2OC)OCO3)cc1F

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.69
TUBB1 Q9H4B7 5/20 0.62
MAPT P10636 6/20 0.56
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
KDM4E B2RXH2 1/20 0.56
NPC1 O15118 1/20 0.56
GAA P10253 1/20 0.56
PKM P14618 1/20 0.56
RAB9A P51151 1/20 0.56
CYP3A4 P08684 4/20 0.53
CYP2D6 P10635 4/20 0.53
CYP2C9 P11712 4/20 0.53
CYP2C19 P33261 4/20 0.53
MCL1 Q07820 1/20 0.53
TUBB4A P04350 2/20 0.52
TUBB P07437 2/20 0.52
TUBA3C P0DPH7 2/20 0.52
TUBA1B P68363 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL997228 1.00 ABCG2 (0.69) ABCG2TUBB1MAPTMEN1KMT2A
SCHEMBL997088 0.93 TUBB1 (0.62) ABCG2TUBB1MAPTMEN1KMT2A
SCHEMBL997089 0.93 TUBB1 (0.62) ABCG2TUBB1MAPTMEN1KMT2A
SCHEMBL996376 0.85 HIF1AN (0.53) ABCG2TUBB1MAPTCYP3A4CYP2D6
SCHEMBL996379 0.85 HIF1AN (0.53) ABCG2TUBB1MAPTCYP3A4CYP2D6
SCHEMBL997900 0.84 MAPT (0.76) ABCG2TUBB1MAPTMEN1KMT2A
SCHEMBL997901 0.84 MAPT (0.76) ABCG2TUBB1MAPTMEN1KMT2A
SCHEMBL998223 0.84 HIF1AN (0.54) ABCG2TUBB1MAPTCYP3A4CYP2D6
SCHEMBL998221 0.84 HIF1AN (0.54) ABCG2TUBB1MAPTCYP3A4CYP2D6
SCHEMBL996848 0.84 TUBB1 (0.76) ABCG2TUBB1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO claimed
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO disclosed