SCHEMBL998221

SCHEMBL998221

COc1ccc(/C=C/C(=O)c2cc3c(cc2OCCN2CCCCC2)OCO3)cc1F

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HIF1AN Q9NWT6 8/20 0.54
ABCG2 Q9UNQ0 1/20 0.51
ACHE P22303 5/20 0.51
BCHE P06276 3/20 0.51
MAOB P27338 2/20 0.49
TUBB1 Q9H4B7 1/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL998223 1.00 HIF1AN (0.54) HIF1ANABCG2ACHEBCHEMAOB
SCHEMBL996376 0.99 HIF1AN (0.53) HIF1ANABCG2ACHEBCHEMAOB
SCHEMBL996379 0.99 HIF1AN (0.53) HIF1ANABCG2ACHEBCHEMAOB
SCHEMBL998195 0.92 HIF1AN (0.54) HIF1ANABCG2TUBB1CYP3A4CYP2D6
SCHEMBL998194 0.92 HIF1AN (0.54) HIF1ANABCG2TUBB1CYP3A4CYP2D6
SCHEMBL998727 0.88 MAPT (0.59) HIF1ANABCG2MAOBTUBB1CYP3A4
SCHEMBL998730 0.88 MAPT (0.59) HIF1ANABCG2MAOBTUBB1CYP3A4
SCHEMBL997108 0.87 MAPT (0.60) HIF1ANABCG2ACHEBCHEMAOB
SCHEMBL997110 0.87 MAPT (0.60) HIF1ANABCG2ACHEBCHEMAOB
SCHEMBL996372 0.86 ACHE (0.52) HIF1ANABCG2ACHEBCHEMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009826-A2 NOVEL CHALCONE DERIVATIVES WITH CYTOTOXIC ACTIVITY ADAMED Sp.z o.o. (PL) 2011-01-27 WO disclosed