SCHEMBL9975265

SCHEMBL9975265

CNc1ccc(OCc2ccc(C)nc2)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 11/20 0.41
KIT P10721 9/20 0.41
FFAR4 Q5NUL3 2/20 0.39
FFAR1 O14842 1/20 0.39
EGFR P00533 1/20 0.39
ERBB2 P04626 1/20 0.39
ERBB3 P21860 1/20 0.39
ERBB4 Q15303 1/20 0.39
APP P05067 2/20 0.37
GAA P10253 1/20 0.37
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
ALOX5 P09917 1/20 0.36
EPHX2 P34913 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28336000 0.86 CSF1R (0.51) CSF1RKITNPC1POLBRAB9A
SCHEMBL6976989 0.86 EGFR (0.45) CSF1RKITEGFRERBB2NPC1
SCHEMBL13814708 0.83 ALDH1A1 (0.47) POLB
SCHEMBL9975354 0.79 PLK1 (0.43) FFAR4ERBB2APPNPC1POLB
SCHEMBL6979978 0.79 FFAR4 (0.54) FFAR4APPL3MBTL1
SCHEMBL6977010 0.77 ERBB2 (0.57) EGFRERBB2ERBB3ERBB4
SCHEMBL22169906 0.76 MAPT (0.51) FFAR4FFAR1GAANPC1RAB9A
SCHEMBL22169907 0.75 MRGPRX4 (0.55) FFAR4
SCHEMBL2250509 0.75 EGFR (0.52) EGFRERBB2ERBB3ERBB4
SCHEMBL6980764 0.73 MRGPRX4 (0.54) EGFRERBB2GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8202879-B2 Quinazoline derivatives having tyrosine kinase inhibitory activity SHIONOGI & CO., LTD. (JP) 2012-06-19 US disclosed
US-20090143414-A1 Quinazoline Derivatives Having Tyrosine Kinase Inhibitory Activity SHIONOGI & CO., LTD. (JP) 2009-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090143414-A1 Quinazoline Derivatives Having Tyrosine Kinase Inhibitory Activity ERBB2, EGFR, ABL1 CSF1R 476/4885KIT 409/4885FFAR4 1426/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.