SCHEMBL9975729

SCHEMBL9975729

CN1CCC(c2cc(I)sc2C(=O)O)=C(C2CCCCC2)C1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.34
PTGS2 P35354 1/20 0.34
HRH1 P35367 1/20 0.34
HTR3A P46098 1/20 0.34
PDE4D Q08499 1/20 0.34
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
ADORA1 P30542 1/20 0.30
RAD52 P43351 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9941462 0.90 ADRA2C (0.33) ADRA2CPTGS2HRH1HTR3APDE4D
SCHEMBL16866368 0.89 TP53 (0.35) ALDH1A1MAPT
SCHEMBL16859522 0.83 ADRA2C (0.38) ADRA2CPTGS2HRH1HTR3APDE4D
SCHEMBL15639028 0.82 ADRA2C (0.39) ADRA2CPTGS2HRH1HTR3APDE4D
SCHEMBL9975863 0.81 MAPT (0.32) KDM4EALDH1A1MAPTADORA1RAD52
SCHEMBL15639462 0.81 NR1I2 (0.41) ADRA2CPTGS2HRH1HTR3APDE4D
SCHEMBL9975903 0.80 MAPT (0.36) ADRA2CPTGS2HRH1HTR3APDE4D
SCHEMBL19397886 0.78 ADRA2C (0.34) ADRA2CPTGS2HRH1HTR3APDE4D
SCHEMBL9975785 0.78 CHRM5 (0.34) MAPT
SCHEMBL10381889 0.75 ADRA2C (0.32) ADRA2CPTGS2HRH1HTR3APDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083105-A1 INHIBITORS OF HEPATITIS C VIRUS POLYMERASE COCRYSTAL DISCOVERY, INC. (US) 2012-06-21 WO disclosed