SCHEMBL9977702

SCHEMBL9977702

O=C(O)C[C@@H]1C2CCC(CC2)C1Nc1nc(-c2n[nH]c3ncc(F)cc23)ncc1F

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 13/20 0.55
GSK3B P49841 13/20 0.55
PIK3CG P48736 11/20 0.54
JAK2 O60674 8/20 0.54
PLK1 P53350 7/20 0.54
PIK3CD O00329 6/20 0.54
PIK3CA P42336 6/20 0.54
ROCK2 O75116 5/20 0.54
ROCK1 Q13464 5/20 0.54
FLT3 P36888 11/20 0.50
SRC P12931 6/20 0.50
PIK3CB P42338 3/20 0.49
PRKACA P17612 5/20 0.48
KDR P35968 4/20 0.48
IRAK4 Q9NWZ3 2/20 0.48
SYK P43405 1/20 0.48
CDK2 P24941 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15400283 1.00 GSK3A (0.55) GSK3AGSK3BPIK3CGJAK2PLK1
SCHEMBL15400279 1.00 GSK3A (0.55) GSK3AGSK3BPIK3CGJAK2PLK1
SCHEMBL15400464 1.00 GSK3A (0.55) GSK3AGSK3BPIK3CGJAK2PLK1
SCHEMBL15400465 1.00 GSK3A (0.55) GSK3AGSK3BPIK3CGJAK2PLK1
SCHEMBL9977673 0.87 GSK3A (0.72) GSK3AGSK3BJAK2FLT3SRC
SCHEMBL9977697 0.87 GSK3A (0.53) GSK3AGSK3BPIK3CGJAK2PLK1
SCHEMBL9940696 0.87 GSK3A (0.72) GSK3AGSK3BJAK2FLT3SRC
SCHEMBL16199093 0.87 GSK3A (0.72) GSK3AGSK3BJAK2FLT3SRC
SCHEMBL16199091 0.87 GSK3A (0.72) GSK3AGSK3BJAK2FLT3SRC
SCHEMBL16199081 0.87 GSK3A (0.72) GSK3AGSK3BJAK2FLT3SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083117-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-21 WO disclosed