SCHEMBL9980375

SCHEMBL9980375

NS(=O)(=O)c1ccc(OCC(F)(F)F)c(CNc2ncnc3[nH]nc(Br)c23)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 8/20 0.40
LMNA P02545 3/20 0.37
BRAF P15056 6/20 0.36
NTRK1 P04629 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CA2 P00918 3/20 0.34
CA1 P00915 2/20 0.34
CA7 P43166 2/20 0.34
CA13 Q8N1Q1 2/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PTGS2 P35354 1/20 0.34
STAT3 P40763 1/20 0.34
PTK2 Q05397 3/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1808559 0.78 TNNI3K (0.62) TNNI3KLMNABRAFALDH1A1CA2
Hydrochloric Acid SCHEMBL1804254 0.77 TNNI3K (0.61) TNNI3KLMNABRAFALDH1A1CA2
SCHEMBL1806158 0.76 BRAF (0.61) TNNI3KLMNABRAFALDH1A1CA2
SCHEMBL1803061 0.76 SMN1; SMN2 (0.46) TNNI3KLMNABRAFSMN1; SMN2ALDH1A1
SCHEMBL12067069 0.76 TNNI3K (0.67) TNNI3KBRAF
SCHEMBL1807400 0.76 TNNI3K (0.55) TNNI3KLMNABRAFALDH1A1CA2
SCHEMBL1806484 0.75 TNNI3K (0.58) TNNI3KBRAFALDH1A1CA2
Hydrochloric Acid SCHEMBL1804510 0.75 BRAF (0.60) TNNI3KLMNABRAFALDH1A1CA2
SCHEMBL9980436 0.75 TNNI3K (0.37) TNNI3KBRAFCA2CA1CA7
SCHEMBL1805541 0.74 BRAF (0.54) TNNI3KLMNABRAFALDH1A1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO claimed
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed