SCHEMBL9980436

SCHEMBL9980436

CN1CCN(c2ccc(S(N)(=O)=O)cc2CNc2ncnc3[nH]nc(Br)c23)CC1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 5/20 0.37
BRAF P15056 4/20 0.37
RAD52 P43351 1/20 0.36
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
CA1 P00915 6/20 0.35
AURKA O14965 1/20 0.35
SOS1 Q07889 1/20 0.34
WDR5 P61964 1/20 0.34
KMT2A Q03164 1/20 0.34
PRKCZ Q05513 1/20 0.34
CA2 P00918 5/20 0.34
CA9 Q16790 3/20 0.34
CA12 O43570 2/20 0.34
CA7 P43166 2/20 0.33
CA13 Q8N1Q1 2/20 0.33
EGFR P00533 1/20 0.33
HRH4 Q9H3N8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9980493 0.90 TNNI3K (0.36) TNNI3KBRAFCA1CA2CA9
SCHEMBL9980424 0.87 TNNI3K (0.35) TNNI3KBRAFCA1CA2CA7
SCHEMBL9980416 0.83 TNNI3K (0.43) TNNI3KBRAFJAK3CA1CA2
SCHEMBL12067033 0.76 TNNI3K (0.62) TNNI3KBRAFWDR5KMT2A
SCHEMBL9980375 0.75 TNNI3K (0.40) TNNI3KBRAFCA1CA2CA7
SCHEMBL9980404 0.74 STK4 (0.39) TNNI3KBRAFKMT2AEGFR
SCHEMBL9980448 0.73 LRRK2 (0.42) TNNI3KBRAFCA1CA2CA9
SCHEMBL9980486 0.71 FFAR2 (0.33) CA1WDR5KMT2ACA2CA7
SCHEMBL1809126 0.68 SRC (0.43) TNNI3KBRAFKMT2AEGFR
SCHEMBL9980393 0.68 TNNI3K (0.40) TNNI3KBRAFCA1CA2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO claimed
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed