SCHEMBL9983380

SCHEMBL9983380

O=C1NC(=O)[C@@]2(COC[C@H]2OCc2ccccc2)N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
CTSV O60911 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
CTSC P53634 1/20 0.36
CTSF Q9UBX1 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
MMP13 P45452 3/20 0.35
MMP2 P08253 2/20 0.35
PSEN1 P49768 4/20 0.34
PSEN2 P49810 4/20 0.34
APH1B Q8WW43 4/20 0.34
NCSTN Q92542 4/20 0.34
APH1A Q96BI3 4/20 0.34
PSENEN Q9NZ42 4/20 0.34
MAPT P10636 2/20 0.34
CYP2C19 P33261 1/20 0.34
MMP14 P50281 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9984914 1.00 ALDH1A1 (0.40) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL9984420 1.00 ALDH1A1 (0.40) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL12023790 0.89 MAPT (0.36) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL9983715 0.88 ALDH1A1 (0.39) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL12024277 0.88 ALDH1A1 (0.39) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL12024360 0.88 ALDH1A1 (0.39) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL13053338 0.80 ALDH1A1 (0.43) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL13053343 0.80 ALDH1A1 (0.43) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL15229601 0.78 TDP1 (0.42) ALDH1A1CTSVCTSLCTSBCTSS
SCHEMBL6239837 0.74 CRBN (0.39) ALDH1A1MAPTLMNACACNA1FCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151348-A1 HETEROCYCLIC AMINO ACIDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-12-08 WO disclosed
WO-2011151348-A1 HETEROCYCLIC AMINO ACIDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-12-08 WO disclosed
EP-2392568-A1 Heterocyclic amino acids for prostate cancer imaging Bayer Pharma Aktiengesellschaft (DE) 2011-12-07 EP disclosed
EP-2392568-A1 Heterocyclic amino acids for prostate cancer imaging Bayer Pharma Aktiengesellschaft (DE) 2011-12-07 EP disclosed