SCHEMBL9985447

SCHEMBL9985447

CNS(=O)(=O)c1ccc(OCC2CCCCC2)c(Nc2[nH]cnc3ncnc2-3)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.47
CDK1 P06493 5/20 0.47
CCNB1 P14635 5/20 0.47
CCNA2 P20248 5/20 0.47
CCNB2 O95067 4/20 0.47
CCNA1 P78396 4/20 0.47
CCNB3 Q8WWL7 4/20 0.47
TNNI3K Q59H18 10/20 0.43
BRD4 O60885 2/20 0.42
CYP19A1 P11511 1/20 0.37
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
CCNT1 O60563 1/20 0.37
ROCK2 O75116 1/20 0.37
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CCNE1 P24864 1/20 0.37
GSK3B P49841 1/20 0.37
CDK7 P50613 1/20 0.37
CDK9 P50750 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9986382 0.91 TNNI3K (0.42) CDK2CDK1CCNB1CCNA2CCNB2
SCHEMBL9986144 0.87 TNNI3K (0.41) CDK2CDK1CCNB1CCNA2CCNB2
SCHEMBL9985709 0.82 TNNI3K (0.45) TNNI3K
SCHEMBL9986569 0.81 TNNI3K (0.45) TNNI3K
SCHEMBL9985780 0.81 TNNI3K (0.43) TNNI3K
SCHEMBL9985668 0.78 TNNI3K (0.44) TNNI3K
SCHEMBL9987082 0.78 TNNI3K (0.43) TNNI3K
SCHEMBL9985735 0.78 TNNI3K (0.46) TNNI3K
SCHEMBL9985716 0.78 TNNI3K (0.56) TNNI3K
SCHEMBL9986214 0.78 TNNI3K (0.50) TNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO claimed
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed