SCHEMBL9986949

SCHEMBL9986949

CCC(Nc1ccc([N+](=O)[O-])c(Nc2ccccc2SC)n1)n1ccnc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.37
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
CYP17A1 P05093 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
CYP19A1 P11511 1/20 0.32
HSF1 Q00613 1/20 0.32
CYP24A1 Q07973 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MAPT P10636 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
NTRK1 P04629 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9985176 0.85 CYP17A1 (0.43) BRD4KMT2AMEN1CYP17A1CYP19A1
SCHEMBL9984879 0.83 BRD4 (0.45) BRD4KMT2AMEN1L3MBTL1CYP19A1
SCHEMBL9984119 0.82 BRD4 (0.44) BRD4KMT2AMEN1CYP19A1HSF1
SCHEMBL9984994 0.81 BRD4 (0.43) BRD4KMT2AMEN1CYP17A1CYP19A1
SCHEMBL9984735 0.80 BRD4 (0.45) BRD4KMT2AMEN1L3MBTL1HSF1
SCHEMBL9985113 0.80 EGFR (0.43) BRD4CYP19A1HSF1MAPT
SCHEMBL9985029 0.80 BRD4 (0.42) BRD4KMT2AMEN1CYP17A1CYP19A1
SCHEMBL9983283 0.80 GAA (0.43) BRD4KMT2AMEN1L3MBTL1CYP19A1
SCHEMBL9984024 0.79 BRD4 (0.41) BRD4CYP19A1HSF1MAPT
SCHEMBL9984037 0.78 BRD4 (0.41) BRD4KMT2ACYP17A1L3MBTL1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394993-A2 NOVEL 2,6-SUBSTITUTED-3-NITROPYRIDINE DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION INCLUDING SAME Dong Wha Pharm. Co., Ltd. (KR) 2011-12-14 EP disclosed