SCHEMBL998713

SCHEMBL998713

N[C@H](C=O)C(C1CCC1)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(Cl)cc2)C1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.53
CYP3A4 P08684 1/20 0.37
RPS6KB1 P23443 2/20 0.33
MAPT P10636 2/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
KIT P10721 1/20 0.31
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1083266 0.88 KCNH2 (0.55) KCNH2CYP3A4
SCHEMBL1001677 0.81 KCNH2 (0.53) KCNH2CYP3A4MAPTPTGDR2TP53
SCHEMBL997860 0.77 KCNH2 (0.58) KCNH2CYP3A4PTGDR2
SCHEMBL998632 0.76 KCNH2 (0.62) KCNH2CYP3A4MAPTTP53GAA
SCHEMBL999072 0.76 KCNH2 (0.51) KCNH2CYP3A4
SCHEMBL2070491 0.76 KCNH2 (0.68) KCNH2CYP3A4MAPTMEN1LMNA
SCHEMBL997258 0.75 KCNH2 (0.65) KCNH2CYP3A4RPS6KB1
SCHEMBL998712 0.75 KCNH2 (0.63) KCNH2CYP3A4MAPTMEN1LMNA
SCHEMBL998298 0.73 KCNH2 (0.54) KCNH2CYP3A4MAPTTP53GAA
SCHEMBL997018 0.73 KCNH2 (0.64) KCNH2CYP3A4MAPTMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451814-A2 FUSED IMIDAZOLES AND COMPOSITIONS COMPRISING THEM FOR THE TREATMENT OF PARASITIC DISEASES, SUCH AS E.G. MALARIA IRM LLC (BM) 2012-05-16 EP claimed
WO-2011006143-A2 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES IRM LLC (BM) 2011-01-13 WO claimed