SCHEMBL9987252

SCHEMBL9987252

CNC(=O)OCn1cc(C(=O)O)c2ccc(Cl)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPT1A P50416 1/20 0.46
CNR1 P21554 2/20 0.40
PRPS1 P60891 1/20 0.40
CNR2 P34972 1/20 0.40
MCL1 Q07820 3/20 0.39
P2RX3 P56373 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CDK2 P24941 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL613579 0.81 CPT1A (0.45) CPT1ACNR1PRPS1CNR2MCL1
SCHEMBL2642676 0.79 KDM4E (0.48) CPT1ACNR1CNR2CA1CA2
SCHEMBL2642993 0.77 CNR2 (0.48) CPT1ACNR1PRPS1CNR2MCL1
SCHEMBL2644030 0.76 CPT1A (0.44) CPT1ACNR1CNR2PTGDR2CA1
SCHEMBL2642659 0.74 CNR2 (0.51) CNR1PRPS1CNR2KDM4EALDH1A1
SCHEMBL3105145 0.74 SERPINE1 (0.59) CPT1ACNR1CNR2CA1CA2
SCHEMBL4660003 0.74 KDM4E (0.48) CPT1ACNR1CNR2KDM4EMEN1
SCHEMBL2643380 0.73 CNR2 (0.56) CNR1CNR2
SCHEMBL3098967 0.73 HTR6 (0.59) CPT1ACNR1PRPS1CNR2MCL1
SCHEMBL612485 0.73 AVPR1A (0.54) CPT1ACNR1CNR2MCL1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2392571-A2 Indol-3-yl-carbonyl-piperidin and piperazin derivatives F. Hoffmann-La Roche AG (CH) 2011-12-07 EP disclosed