SCHEMBL9988152

SCHEMBL9988152

O=C(O)C1CCN(c2ccc(Nc3nc(N4CCC(O)CC4)ccc3[N+](=O)[O-])cc2F)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
SERPINE1 P05121 6/20 0.44
MAPT P10636 5/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
JAK2 O60674 1/20 0.39
BRD4 O60885 1/20 0.39
GAA P10253 1/20 0.39
RHOA P61586 1/20 0.39
PDE7A Q13946 2/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9984012 0.94 MAPT (0.47) TDP1MAPTKMT2AMEN1ALDH1A1
SCHEMBL9983927 0.92 MAPT (0.49) TDP1MAPTKMT2AMEN1ALDH1A1
SCHEMBL9987975 0.91 FLT3 (0.46) TDP1SERPINE1MAPTKMT2AMEN1
SCHEMBL9983445 0.90 ALDH1A1 (0.45) TDP1MAPTKMT2AMEN1ALDH1A1
SCHEMBL9984347 0.89 MAPT (0.43) TDP1MAPTKMT2AMEN1ALDH1A1
SCHEMBL9984527 0.89 MAPT (0.43) TDP1MAPTKMT2AMEN1ALDH1A1
SCHEMBL9984987 0.89 MAPT (0.42) TDP1MAPTKMT2AMEN1ALDH1A1
SCHEMBL9984266 0.89 CDK4 (0.43) MAPTKMT2AMEN1ALDH1A1POLB
SCHEMBL9984594 0.89 CDK4 (0.43) MAPTKMT2AMEN1ALDH1A1POLB
SCHEMBL9984020 0.89 FLT3 (0.46) MAPTKMT2AMEN1ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394993-A2 NOVEL 2,6-SUBSTITUTED-3-NITROPYRIDINE DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION INCLUDING SAME Dong Wha Pharm. Co., Ltd. (KR) 2011-12-14 EP disclosed