SCHEMBL9988166

SCHEMBL9988166

CC(N)c1cnc(OCCF)c(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.34
HTR2C P28335 3/20 0.34
PIK3CA P42336 1/20 0.33
MTOR P42345 1/20 0.33
S1PR1 P21453 3/20 0.32
AAK1 Q2M2I8 3/20 0.32
IDH1 O75874 5/20 0.32
CYP17A1 P05093 1/20 0.32
SCN9A Q15858 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15599195 0.88 IDH1 (0.33) HTR2AHTR2CAAK1IDH1CYP17A1
Hydrochloric Acid SCHEMBL15351153 0.83 IDH1 (0.34) HTR2APIK3CAMTORAAK1IDH1
SCHEMBL13877375 0.83 S1PR1 (0.38) S1PR1AAK1SCN9A
SCHEMBL18266454 0.82 SCN9A (0.34) S1PR1AAK1SCN9A
SCHEMBL4550399 0.82 SCN9A (0.39) S1PR1SCN9A
Hydrochloric Acid SCHEMBL4225843 0.81 S1PR1 (0.38) S1PR1AAK1SCN9A
Hydrochloric Acid SCHEMBL27777869 0.81 S1PR1 (0.38) S1PR1AAK1SCN9A
SCHEMBL4550317 0.81 IDH1 (0.43) AAK1IDH1CYP17A1SCN9A
SCHEMBL16045149 0.81 IDH1 (0.43) AAK1IDH1CYP17A1SCN9A
SCHEMBL9988673 0.81 RORC (0.37) PIK3CAMTORS1PR1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966156-B1 NEW COMPOUNDS III ASTRAZENECA AB (SE) 2011-12-21 EP disclosed