SCHEMBL9989772

SCHEMBL9989772

NC(=O)c1cc(Cl)cc2[nH]c(-c3ccc(C4CCCN4C(=O)O)cc3)nc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.65
PARP2 Q9UGN5 8/20 0.57
MAP4K4 O95819 1/20 0.51
INSR P06213 1/20 0.51
CSF1R P07333 1/20 0.51
PIM1 P11309 1/20 0.51
FLT4 P35916 1/20 0.51
FLT3 P36888 1/20 0.51
CLK2 P49760 1/20 0.51
IRAK1 P51617 1/20 0.51
ITK Q08881 1/20 0.51
MAP4K2 Q12851 1/20 0.51
DYRK1A Q13627 1/20 0.51
PIM3 Q86V86 1/20 0.51
MINK1 Q8N4C8 1/20 0.51
AURKB Q96GD4 1/20 0.51
HIPK2 Q9H2X6 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
MKNK2 Q9HBH9 1/20 0.51
ALK Q9UM73 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4969641 0.88 PARP1 (0.59) PARP1PARP2MAP4K4INSRCSF1R
SCHEMBL4968077 0.88 PARP1 (0.74) PARP1PARP2MAP4K4INSRCSF1R
SCHEMBL4971299 0.86 PARP1 (0.64) PARP1PARP2MAP4K4INSRCSF1R
SCHEMBL9989160 0.85 PARP1 (0.77) PARP1PARP2DHODH
SCHEMBL4971493 0.85 PARP1 (0.75) PARP1PARP2MAP4K4INSRCSF1R
SCHEMBL4971182 0.80 PARP1 (0.73) PARP1PARP2MAP4K4INSRCSF1R
SCHEMBL4970604 0.79 PARP1 (1.00) PARP1PARP2MAP4K4INSRCSF1R
SCHEMBL4972871 0.78 PARP1 (0.72) PARP1PARP2MAP4K4INSRCSF1R
SCHEMBL4973364 0.78 MAP4K4 (0.76) PARP1PARP2MAP4K4INSRCSF1R
SCHEMBL4968533 0.76 PARP1 (0.74) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038751-A3 PROCESS FOR THE PURIFICATION OF AROMATIC DICARBOXYLIC ACID DAVY PROCESS TECHNOLOGY LIMITED (GB) 2012-05-10 WO disclosed
EP-1957477-B1 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH PHENYL AT THE 2-POSITION ARE POTENT PARP INHIBITORS ABBOTT LAB (US) 2011-12-07 EP disclosed