SCHEMBL9992

SCHEMBL9992

CCOC(=O)C1(c2ccc(-c3ccccc3-c3onc(C)c3Nc3cccc(-c4cccc(F)c4OC)n3)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC3 O15438 1/20 0.36
ABCC4 O15439 1/20 0.36
ABCB11 O95342 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2C9 P11712 1/20 0.36
ABCB4 P21439 1/20 0.36
LPAR1 Q92633 1/20 0.36
ABCC2 Q92887 1/20 0.36
SLCO1B3 Q9NPD5 1/20 0.36
SLCO1B1 Q9Y6L6 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA5A P35218 1/20 0.35
CA9 Q16790 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
ADORA2A P29274 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4512 0.95 ABCC3 (0.40) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL9991 0.94 LMNA (0.35) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL10210 0.92 ABCC3 (0.40) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL10568 0.92 LPAR1 (0.44) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL4921 0.88 ABCC3 (0.44) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL9784 0.88 ABCC3 (0.42) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL4494 0.87 LPAR1 (0.44) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL4640 0.86 ABCC3 (0.41) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL10209 0.86 LMNA (0.36) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL4079 0.85 LPAR1 (0.49) ABCC3ABCC4ABCB11CYP2C8CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed