SCHEMBL10018183

SCHEMBL10018183

COc1ccc2c3c(cc(O)c2c1)C(C)(C)C(C)(O)c1ccccc1-3

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
PDK2 Q15119 6/20 0.41
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HSP90AA1 P07900 1/20 0.34
PARP1 P09874 1/20 0.34
AR P10275 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC4 P56524 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
CDK1 P06493 2/20 0.33
CCNB1 P14635 2/20 0.33
GSK3B P49841 2/20 0.33
POLB P06746 1/20 0.33
CCNB2 O95067 1/20 0.33
GSK3A P49840 1/20 0.33
CDK5 Q00535 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10018176 0.92 MEN1 (0.44) GAAMEN1KMT2APDK2MAPT
SCHEMBL8513625 0.86 MEN1 (0.43) GAAMEN1KMT2APDK2MAPT
SCHEMBL14046448 0.84 PDK2 (0.36) GAAMEN1KMT2APDK2MAPT
SCHEMBL10018205 0.82 MEN1 (0.39) GAAMEN1KMT2APDK2HSP90AA1
SCHEMBL9898233 0.82 MEN1 (0.45) GAAMEN1KMT2APDK2MAPT
SCHEMBL3947184 0.81 KMT2A (0.42) GAAMEN1KMT2APDK2HSP90AA1
SCHEMBL10018210 0.81 MEN1 (0.40) GAAMEN1KMT2APDK2HSP90AA1
SCHEMBL12424597 0.81 PDK2 (0.42) GAAMEN1KMT2APDK2ALDH1A1
SCHEMBL10018179 0.81 GAA (0.38) GAAMEN1KMT2APDK2MAPT
SCHEMBL9932428 0.81 MEN1 (0.43) GAAMEN1KMT2APDK2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8123987-B2 Chromene compounds TOKUYAMA CORPORATION (JP) 2012-02-28 US disclosed
US-8123987-B2 Chromene compounds TOKUYAMA CORPORATION (JP) 2012-02-28 US disclosed
US-20100230648-A1 Chromene Compounds TOKUYAMA CORPORATION (JP) 2010-09-16 US disclosed
US-20100230648-A1 Chromene Compounds TOKUYAMA CORPORATION (JP) 2010-09-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100230648-A1 Chromene Compounds H1-4, RB1, H1-0 GAA 4225/4885MEN1 1057/4885KMT2A 269/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.